Cetrorelix Acetate CAS 130143-01-0 GnRH antagonist Peptide Tsarkake (HPLC) ≥98.0% Babban inganci
Shanghai Ruifu Chemical Co., Ltd. shine babban kamfani na Cetrorelix Acetate (CAS: 130143-01-0) tare da babban inganci.Cetrorelix Acetate shine hormone mai sakin gonadotropin (GnRH).Ruifu Chemical yana ba da jerin GMP peptides.Ruifu na iya samar da isar da saƙo na duniya, farashi mai gasa, ƙanana da yawa da ake samu.Sayi Cetrorelix Acetate,Please contact: alvin@ruifuchem.com
Sunan Sinadari | Cetrorelix acetate |
Makamantu | N-Acetyl-3-(2-Naphthalenyl)-D-Alanyl-4-Chloro-D-Phenylalanyl-3-(3-Pyridinyl)-D-Alanyl-L-Seryl-L-Tyrosyl-N5-(Aminocarbonyl)- D-Ornithyl-L-Leucyl-L-Arginyl-L-Prolyl-D-Alaninamide Diacetate;NS-75A Diacetate;Saukewa: SB-075 |
Jeri | Ac-3-(2-naphthyl) -D-Ala-4-Chloro-D-Phe-3(3-pyridyl)-D-Ala-Ser-Tyr-D-Cit-Leu-Arg-Pro-D-Ala -NH2 |
Lambar CAS | 130143-01-0 |
Matsayin Hannun jari | A cikin Hannun jari, Ma'aunin Samarwa Har zuwa Kilogram |
Tsarin kwayoyin halitta | Saukewa: C70H92N17O14 |
Nauyin Kwayoyin Halitta | 1551.16 |
Adana Yanayin. | Wuri mai sanyi & bushewa (-20 ℃).Firiji |
Rayuwar Rayuwa | >Shekaru 2 Idan An Ajiyesu Da Kyau |
Kashi | GMP Peptides |
Takardu | COA, MS, HPLC, NMR, MSDS, da dai sauransu. |
Alamar | Ruifu Chemical |
Abu | Ƙayyadaddun bayanai |
Bayyanar | Farin Foda |
Peptide Tsabta (na HPLC) | ≥98.0% (ta Haɗin Yanki) |
Abun cikin Peptide | ≥80.0% (ta %N) |
Amino Acid Haɗin Kai | 10% na Theetical |
Abun ciki na Acetate | ≤10.0% (na HPLC) |
Abubuwan ciki na TFA | ≤1.0% |
Tsaftace Guda Daya | ≤1.0% (na HPLC) |
Abubuwan Ruwa (Karl Fischer) | ≤8.0% |
Assay | 95.0 ~ 105.0% (Ta Anhydrous, Acetic Acid-Free) |
MS | Daidaitawa |
Matsayin Gwaji | Matsayin Kasuwanci |
Bukatun jigilar kaya | Jakunkuna na Kankara, Jakunkuna na Desiccant |
Asalin samfur | Na roba |
Hankali | Don Bincike kawai, Ba don amfanin ɗan adam ba |
Amfani | Maganin roba na GnRH Receptor |
Kunshin:Filayen filastik (wanda aka keɓe don tattarawar peptide) ko gilashin gilashi, adadi gwargwadon buƙatun abokin ciniki.
Yanayin Ajiya:Ajiye a cikin kwantena da aka rufe a wurin sanyi da bushe (2 ~ 8 ℃) nesa da abubuwan da ba su dace ba.Kare daga haske da danshi.
Jirgin ruwa:Bayarwa ga duniya ta FedEx / DHL Express.Bayar da isarwa cikin sauri kuma abin dogaro.
Cetrorelix Acetate (CAS 130143-01-0) antagonist ne mai sakin gonadotropin (GnRH) wanda aka sayar da farko a ƙarƙashin sunan alamar Cetrotide.Ana amfani da decapeptide na roba, ana amfani da shi a cikin taimakon haifuwa don hana hawan hormone luteinizing wanda bai kai ba.Da miyagun ƙwayoyi yana aiki ta hanyar toshe aikin GnRH akan pituitary, don haka da sauri yana hana samarwa da aikin luteinizing hormone (LH) da kuma follicle-stimulating hormone (FSH).Cetrorelix Acetate ya ƙunshi nau'o'in amino acid waɗanda ba na halitta ba waɗanda ke hana ovulation da wuri a cikin gwaje-gwajen asibiti, wanda ke haifar da tarin ovulation da kuma taimakon fasahar haifuwa ga marasa lafiya da ke jujjuyawar kwai.
Nuna Cetrorelix Acetate wani hormone ne na wucin gadi wanda ke toshe tasirin hormone mai sakin gonadotropin (GnRH).A cikin fasahar haifuwa da aka taimaka, a cikin marasa lafiya tare da sarrafa kuzarin kwai, hana ovulation da wuri.
Ayyukan Pharmacological Cetrorelix Acetate shine antagonist mai sakin gonadotropin (GnRH).GnRH na iya ɗaure ga masu karɓar membrane na sel pituitary.Cetrorelix acetate gasa yana ɗaure ga waɗannan masu karɓa tare da GnRH na endogenous, ta haka kashi-dogara yana hana ɓoyewar hormone luteinizing (LH) da hormone mai haɓakawa (FSH) ta hanyar adenohypophysis.An haifar da tasirin hanawa nan da nan bayan gudanar da cetrorelix acetate, kuma ana iya kiyaye tasirin hanawa ta hanyar ci gaba da jiyya.ga mata, Cetrorelix Acetate na iya jinkirta kololuwar LH, ta haka jinkirta ovulation.Ga matan da ke fama da motsa jiki na ovarian, tsawon lokacin aikin ya dogara da kashi.An kiyasta kashi ɗaya na cetrorelix 3mg don samun sakamako mai hanawa na akalla kwanaki 4, tare da tasirin hanawa na kusan 70% a ranar 4. Maimaita gudanarwa na cetrorelix acetate 0.25mg kowane sa'o'i 24 zai iya kula da tasirinsa.Sakamakon hormone-antagonizing na Cetrorelix Acetate ya juya gaba daya a ƙarshen jiyya a cikin dabbobi da mutane.
Ayyukan Halittu Cetrorelix Acetate babban mai adawa ne na mai karɓar GnRH tare da ƙimar IC50 na 1.21 nM.
Manufar IC50: 1.21 nM GnRH.