Sitagliptin CAS 486460-32-6 Ma'ema'e >99.0% (HPLC) API Hale Hana Ma'ema'e Ki'eki'e
Hoʻolako i nā mea kikowaena pili i ka Sitagliptin Phosphate Monohydrate:
Sitagliptin API CAS 486460-32-6
Sitagliptin Phosphate Monohydrate API CAS 654671-77-9
2,4,5-Trifluorophenylacetic Acid CAS 209995-38-0
Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Butyric Acid CAS 486460-00-8
Sitagliptin Triazole Hydrochloride CAS 762240-92-6
Sitagliptin Phosphate Monohydrate Intermediate CAS 486460-21-3
Inoa Kimia | ʻO Sitagliptin |
Nā huaʻōlelo like | (3R)-3-Amino-1-[3-(trifluoromethyl)-5,6,7,8-tetrahydro-1,2,4-triazolo[4,3-a]pyrazin-7-yl]-4- (2,4,5-trifluorophenyl)butan-1-kahi |
Helu CAS | 486460-32-6 |
Kūlana Kūʻai | Ma ka waihona, hoʻonui ʻia a hiki i nā tona |
ʻĀpana Molekala | C16H15F6N5O |
Kaumaha Molecular | 407.31 |
Lae hehee | 114.0~115.0 ℃ |
Brand | Kemika Ruifu |
'ikamu | Nā kikoʻī |
Ka nana aku | Keʻokeʻo a i ka pauka kristal keʻokeʻo |
ʻIke ʻia e HPLC | ʻO ka manawa paʻa o ka laʻana e kūlike me ka maʻamau kuhikuhi |
Nalo ma ka maloo | <1.0% |
Koena ma ka Ignition | <0.20% |
Na mea pili | |
ʻO kēlā me kēia haumia hoʻokahi | <0.50% |
Huina paumaele | <1.0% |
Maemae | >99.0% (HPLC) |
Maʻemaʻe Enantiomeric | <0.50% |
Nā Metala Kaumaha | <20ppm |
Kūlana hoʻāʻo | Kūlana ʻoihana |
Hoʻohana | API;Type II Diabetes Mellitus |
Pūʻolo: ʻO ka ʻōmole, ʻeke ʻeke alumini, 25kg / pahu pahu pahu, a i ʻole e like me ka makemake o ka mea kūʻai aku.
Kūlana mālama:E mālama i loko o nā pahu i hoʻopaʻa ʻia ma kahi maloʻo a maloʻo;E pale i ka malamalama a me ka wai.
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ʻO Sitagliptin (CAS: 486460-32-6), ma ke ʻano he ʻano lāʻau antidiabetic hou, ʻo Sitagliptin Phosphate ka mea maikaʻi o ka hilinaʻi glucose, ka hopena hypoglycemic haʻahaʻa, hoʻonui i ka huna me ka hypoglycemia, hoʻopau maikaʻi i ka pōloli, a ʻaʻohe hopena ʻaoʻao e like me ka nausea, luaʻi, edema a hoʻonui i ke kaumaha o ke kino.ʻO Sitagliptin phosphate ma ke ʻano he lāʻau lapaʻau hoʻokahi i nā mea maʻi me ka maʻi diabetes type II hiki ke hōʻemi nui i ka pae o ka hemoglobin glycosylated (HbA1c).ʻO ia ka dipeptidyl peptidase-4 (DPP-4) inhibitor, hiki ke hoʻomaikaʻi i ke kino o ke kanaka e hōʻemi i ke kiʻekiʻe o ka glucose koko.Ua hoʻomohala ʻia ʻo Sitagliptin e Merck & Co. a ʻae ʻia no ka hoʻohana lāʻau lapaʻau ma ʻAmelika Hui Pū ʻIa i ka makahiki 2006.
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Sitagliptin CAS 486460-32-6 Maʻemaʻe >99.0% (HPLC...
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Sitagliptin Phosphate Monohydrate CAS 654671-77...
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2,4,5-Trifluorophenylacetic Acid CAS 209995-38-...
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Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Buty...
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Sitagliptin Triazole Hydrochloride CAS 762240-9...
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ʻO Sitagliptin Phosphate Monohydrate Intermediate ...