Sitagliptin CAS 486460-32-6 Purity > 99.0% (HPLC) API Hoobkas High Purity
Muab Sitagliptin Phosphate Monohydrate Related Intermediates:
Sitagliptin API CAS 486460-32-6
Sitagliptin Phosphate Monohydrate API CAS 654671-77-9
Tom ntej: 2,4,5-Trifluorophenylacetic Acid CAS 209995-38-0
Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Butyric Acid CAS 486460-00-8
Sitagliptin Triazole Hydrochloride CAS 762240-92-6
Sitagliptin Phosphate Monohydrate Intermediate CAS 486460-21-3
Tshuaj npe | Sitagliptin |
Synonyms | (3R)-3-Amino-1-[3-(trifluoromethyl)-5,6,7,8-tetrahydro-1,2,4-triazolo[4,3-a]pyrazin-7-yl]-4- (2,4,5-trifluorophenyl)butan-1-ib |
CAS Nr | 486460-32-6 |
Tshuag xwm txheej | Nyob rau hauv Tshuag, ntau lawm Scale mus txog Tons |
Molecular Formula | C16H15F6N5O |
Molecular Luj | 407.31 Nws |
Melting Point | 114.0 ~ 115.0 ℃ |
Hom | Ruifu Tshuaj |
Yam khoom | Specifications |
Qhov tshwm sim | Dawb rau Off-White Crystalline Hmoov |
Kev txheeb xyuas los ntawm HPLC | Lub Sijhawm khaws cia ntawm Cov Qauv yog Concordant Nrog Reference Standard |
Poob rau ziab | <1.0% |
Residue ntawm Ignition | <0.20% |
Yam khoom muaj feem | |
Ib qho Impurity | <0.50% |
Tag nrho cov impurities | <1.0% |
Purity | > 99.0% (HPLC) |
Enantiomeric Purity yog qhov zoo | <0.50% |
Hnyav Hlau | <20 ppm |
Test Standard | Enterprise Standard |
Kev siv | API;Hom II Mob ntshav qab zib mellitus |
Pob: Lub raj mis, Aluminium ntawv ci hnab, 25kg / Cardboard Nruas, los yog raws li tus neeg yuav tsum tau muaj.
Cia txias:Khaws rau hauv cov thawv ntim khoom ntawm qhov chaw txias thiab qhuav;Tiv thaiv los ntawm lub teeb thiab noo noo.
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Sitagliptin (CAS: 486460-32-6), raws li hom tshiab ntawm cov tshuaj tiv thaiv kab mob ntshav qab zib, Sitagliptin Phosphate muaj qhov zoo ntawm cov piam thaj, cov nyhuv hypoglycemic nruab nrab, nce secretion tsis muaj hypoglycemia, txo qis kev tshaib kev nqhis, thiab tsis muaj kev phiv xws li xeev siab, ntuav, edema thiab nce lub cev hnyav.Sitagliptin phosphate ua ib qho tshuaj kho mob rau cov neeg mob ntshav qab zib hom II tuaj yeem txo qis glycosylated hemoglobin (HbA1c).Nws yog dipeptidyl peptidase-4 (DPP-4) inhibitor, uas tuaj yeem txhim kho tib neeg lub cev lub peev xwm los txo cov ntshav qabzib siab.Sitagliptin tau tsim los ntawm Merck & Co. thiab tau pom zoo rau kev siv kho mob hauv Tebchaws Meskas hauv xyoo 2006.
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Sitagliptin CAS 486460-32-6 Purity > 99.0% (HPLC ...
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Sitagliptin Phosphate Monohydrate CAS 654671-77 ...
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2,4,5-Trifluorophenylacetic Acid CAS 209995-38-...
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Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Buty...
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Sitagliptin Triazole Hydrochloride CAS 762240-9 ...
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Sitagliptin Phosphate Monohydrate Intermediate ...