Tacrolimus FK-506 Fujimycin CAS 104987-11-3 API wheketere parakore teitei
Kaihanga me te Pure Nui me te Kounga Pumau
Ingoa matū: Tacrolimus
Nga kupu taurite: FK-506;Fujimycin
CAS: 104987-11-3
API, Kounga Teitei, Hanganga Aromoni
Ingoa matū | Tacrolimus |
Nga kupu taurite | FK-506;Fujimycin |
Tau CAS | 104987-11-3 |
Tau CAT | RF-API46 |
Tūnga Taonga | I roto i te Stock, Production Tauine Up ki Taranata |
Tātai rāpoi | C44H69NO12 |
Taumaha rāpoi | 804.02 |
Waitohu | Ruifu Chemical |
Tūemi | Whakatakotoranga |
Te ahua | Paura Paa-ma-ma-ma-ma-ma-ma-ma ranei, Kowhai Kowhai Paera Pai, Kare he kakara, he reka reka motuhake |
Tautuhinga | Me Tauhohenga Pai |
Maramatanga | Kia mau ki te Paerewa |
pH | 5.0~6.0 |
pūhaumāota | ≤0.014% |
pūkawa | ≤0.029% |
Konga Taamaha (Pb) | ≤10ppm |
Arsenic | ≤0.0002% |
makuku (KF) | ≤8.0% |
Te toenga i runga i te mura | 18.0%~22.0% |
Te whakamatautau | ≥72.0% (HPLC, i runga i te whakamaroke) |
Paerewa Whakamatau | Paerewa hinonga |
Whakamahinga | API |
Mōkī: Pounamu, Peeke konumohe konumohe, Pahu Kaata, 25kg / Drum, kia rite ranei ki te hiahia a te kaihoko.
Tikanga Rokiroki:Whakaorangia i roto i nga ipu kua hiri ki te waahi makariri me te maroke;Whakaorangia mai i te marama, te makuku me te mate kino.
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Ko te Tacrolimus (he FK-506, Fujimycin ranei) he rongoa whakangao i te mate o te tinana i muri i te whakawhitinga okana ki te whakaiti i te mahi o te punaha mate o te manawanui, me te tupono ki te aukati okana.Ka whakamahia ano hoki i roto i te whakareri i runga i te waahi mo te maimoatanga o te mate mate pukupuku nui, te uveitis kino kino i muri i te whakawhitinga o te hinu wheua, me te mate kiri vitiligo.I tangohia tuatahi a Tacrolimus mai i te hupa FERMENTATION a Streptomyces tsukuba, he moroiti oneone i kitea i Tsukuba, Japan.I ahu mai te ingoa tacrolimus ma te tango i te 't' mo Tsukuba, te ingoa o te maunga i tangohia ai te tauira oneone, 'acrol' mo te macrolide me te 'imus' mo te immunosuppressant.Ahakoa te hangahanga kore e hono ki te cyclosporin, he rite tonu te ahua o te tacrolimus o nga paanga immunosuppressive ki tenei kaihoko i te taumata pūkoro me te molecular.Ko nga rangahau tuatahi i tohu ko te tacrolimus he immunosuppressant kaha, e whakaatu ana i te 100-nui ake te kaha in vitro nui atu i te cyclosporin hei aukati i te whakahohenga o te pūtau T.I muri mai i roto i nga rangahau vivo kua kitea te whai hua o te tacrolimus ki te pehi i te mate autoimmune ohorere me te whakamatautau, me te aukati i te aukati allograft me te xenograft i roto i nga tauira kararehe o te whakawhitinga okana.I te tuatahi, i whakamahia te tacrolimus mo te aukati i te mate o nga turoro kua pa ki te whakawhitinga allograft hei aukati i a raatau ki te whakakore i o raatau mahi hou.Heoi, i muri tata mai, na te painga o te puiao, i kitea ka taea e te tacrolimus te whakaputa hua pai mo nga mate kiri o etahi o nga turoro i tukuna i te whakawhitinga.Na te kitenga o te tacrolimus ka nui ake te maarama ki te mate kiri, hei tauira mo te mate mate pukupuku.I muri mai, i panuitia etahi atu tono mo te tacrolimus me te whakamahi i tenei kaihoko i roto i te dermatology kei te piki haere.
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