Tolvaptan CAS 150683-30-0 API Pure >99.0% (HPLC)

Whakaahuatanga Poto:

Ingoa matū: Tolvaptan

CAS: 150683-30-0

Pure (HPLC): >99.0%

Te ahua: Ma ki te Paura Tioataata-Ma

He kaitukino kaha me te kowhiria te kaikawe kaikawe vasopressin V2

API Kounga Teitei, Hanganga Tauhokohoko

Inquiry: alvin@ruifuchem.com  


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Whakaahuatanga:

Ngā Āhuatanga matū:

Ingoa Tolvaptan
Ingoa matū N-[4-(9-chloro-6-hydroxy-2-azabicyclo[5.4.0]undeca-8,10,12-triene-2-carbonyl)-3-methyl-phenyl]-2-methyl-benzamide
Tau CAS 150683-30-0
Tau CAT RF-API101
Tūnga Taonga I roto i te Stock, Production Tauine Up ki Taranata
Tātai rāpoi C26H25ClN2O3
Taumaha rāpoi 448.94
Waitohu Ruifu Chemical

Whakatakotoranga:

Tūemi Whakatakotoranga
Te ahua Ma ki te Paura Tioata-White
Nga Tikanga Tautuhi IR, HPLC
Wairewa Wairewa i roto i te Benzyl Alcohol me te Methanol engari Tino Karekau i te Wai me te Hexane
Te Maama / Tikanga Tatauria >99.0% (HPLC)
Iwi Whakarewa 219.0~222.0 ℃
Ngaronga i te whakamaroke <0.50%
Te toenga i runga i te mura <0.10%
Te poke kotahi <0.50%
Nga poke katoa <1.00%
Nga Korewa Taamaha ≤20ppm
Wairewa toenga Tutaki ki te Whakatakotoranga
Paerewa Whakamatau Paerewa hinonga
Whakamahinga API;Takawaenga Rongoa

Mōkī me te Rokiroki:

Mōkī: Pounamu, Peeke konumohe konumohe, 25kg / Kaata Drum, kia rite ranei ki te hiahia a te kaihoko

Tikanga Rokiroki:Whakaorangia i roto i nga ipu kua hiri ki te waahi makariri me te maroke;Tiaki i te marama me te makuku

Painga:

1

FAQ:

Taupānga:

Ko Tolvaptan (CAS: 150683-30-0), e mohiotia ana ano ko OPC-41061, he kaitukino, he whakataetae arginine vasopressin receptor 2 antagonist i whakamahia ki te hamani i te hyponatremia (nga taumata konutai toto iti) e pa ana ki te ngoikore o te ngakau, cirrhosis, me te mate o te mate. kore tika te taiaki antidiuretic (SIADH).Otsuka Pharmaceutical tolvaptan raihana i raro i te ingoa hokohoko Samsca i muri i te whakaaetanga a te FDA i te tarukino i Mei 2009. Kua whakaatu ano a Tolvaptan i te kaha ki te mate pukupuku polycystic.I roto i te whakamatautauranga o te tau 2004, ko te tolvaptan i whakahaerehia me nga diuretics tuku iho i tohuhia ki te whakanui ake i te whakahekenga o te nui o te wai me te whakapai ake i nga taumata konutai toto i roto i nga turoro me te ngoikore o te ngakau me te kore e whakaputa i nga paanga kino penei i te hypotension (te whakaheke toto) me te hypokalemia (te whakaheke i nga taumata toto o te pāhare pāporo).Ko te rongoa hoki kaore he paanga kino ki te mahi whatukuhu.

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