Tolvaptan CAS 150683-30-0 API Pure >99.0% (HPLC)
Kaihanga Kaihanga Tolvaptan me nga Takawaenga Paanga:
Tolvaptan CAS 150683-30-0
7-Chloro-1,2,3,4-tetrahydrobenzo[b]azepin-5-one CAS 160129-45-3
o-Toluoyl Chloride CAS 933-88-0
4-Amino-2-Methylbenzoic Acid CAS 2486-75-1
2-Methyl-4-Nitrobenzoic Waikawa CAS 1975-51-5
Ingoa | Tolvaptan |
Ingoa matū | N-[4-(9-chloro-6-hydroxy-2-azabicyclo[5.4.0]undeca-8,10,12-triene-2-carbonyl)-3-methyl-phenyl]-2-methyl-benzamide |
Tau CAS | 150683-30-0 |
Tau CAT | RF-API101 |
Tūnga Taonga | I roto i te Stock, Production Tauine Up ki Taranata |
Tātai rāpoi | C26H25ClN2O3 |
Taumaha rāpoi | 448.94 |
Waitohu | Ruifu Chemical |
Tūemi | Whakatakotoranga |
Te ahua | Ma ki te Paura Tioata-White |
Nga Tikanga Tautuhi | IR, HPLC |
Wairewa | Wairewa i roto i te Benzyl Alcohol me te Methanol engari Tino Karekau i te Wai me te Hexane |
Te Maama / Tikanga Tatauria | >99.0% (HPLC) |
Iwi Whakarewa | 219.0~222.0 ℃ |
Ngaronga i te whakamaroke | <0.50% |
Te toenga i runga i te mura | <0.10% |
Te poke kotahi | <0.50% |
Nga poke katoa | <1.00% |
Nga Korewa Taamaha | ≤20ppm |
Wairewa toenga | Tutaki ki te Whakatakotoranga |
Paerewa Whakamatau | Paerewa hinonga |
Whakamahinga | API;Takawaenga Rongoa |
Mōkī: Pounamu, Peeke konumohe konumohe, 25kg / Kaata Drum, kia rite ranei ki te hiahia a te kaihoko
Tikanga Rokiroki:Whakaorangia i roto i nga ipu kua hiri ki te waahi makariri me te maroke;Tiaki i te marama me te makuku
![1](https://a395.goodao.net/uploads/15.jpg)
![](https://a395.goodao.net/uploads/23.jpg)
Ko Tolvaptan (CAS: 150683-30-0), e mohiotia ana ano ko OPC-41061, he kaitukino, he whakataetae arginine vasopressin receptor 2 antagonist i whakamahia ki te hamani i te hyponatremia (nga taumata konutai toto iti) e pa ana ki te ngoikore o te ngakau, cirrhosis, me te mate o te mate. kore tika te taiaki antidiuretic (SIADH).Otsuka Pharmaceutical tolvaptan raihana i raro i te ingoa hokohoko Samsca i muri i te whakaaetanga a te FDA i te tarukino i Mei 2009. Kua whakaatu ano a Tolvaptan i te kaha ki te mate pukupuku polycystic.I roto i te whakamatautauranga o te tau 2004, ko te tolvaptan i whakahaerehia me nga diuretics tuku iho i tohuhia ki te whakanui ake i te whakahekenga o te nui o te wai me te whakapai ake i nga taumata konutai toto i roto i nga turoro me te ngoikore o te ngakau me te kore e whakaputa i nga paanga kino penei i te hypotension (te whakaheke toto) me te hypokalemia (te whakaheke i nga taumata toto o te pāhare pāporo).Ko te rongoa hoki kaore he paanga kino ki te mahi whatukuhu.