2,4,5-Trifluorophenylacetic Acid CAS 209995-38-0 Purità ≥99.5% (GC) Sitagliptin Phosphate Monohydrate Intermedju
Provvista Sitagliptin Phosphate Monohydrate Intermedji Relatati:
Sitagliptin API CAS 486460-32-6
Sitagliptin Phosphate Monohydrate API CAS 654671-77-9
Aċidu 2,4,5-trifluworofenilaċetiku CAS 209995-38-0
Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Butyric Acid CAS 486460-00-8
Sitagliptin Triazole Hydrochloride CAS 762240-92-6
Sitagliptin Phosphate Monohydrate Intermedju CAS 486460-21-3
Isem Kimiku | Aċidu 2,4,5-Trifluorofenilaċetiku |
Numru CAS | 209995-38-0 |
Numru tal-KAT | RF-PI1191 |
Status tal-istokk | Fil-Ħażna, Skala ta' Produzzjoni Sa Tunnellati |
Formula Molekulari | C8H5F3O2 |
Piż Molekulari | 190.12 |
Punt tat-tidwib | 121.0 sa 125.0 ℃ |
Solubilità | Solubbli fil-Metanol |
Brand | Ruifu Kimika |
Oġġett | Speċifikazzjonijiet |
Dehra | Trab abjad għal Off-White |
Purità / Metodu ta 'Analiżi | ≥99.5% (GC) |
Umdità (KF) | ≤0.50% |
Residwu fuq Igniton | ≤0.50% |
Impuritajiet Totali | ≤0.50% |
Standard tat-Test | Standard tal-Intrapriża |
Użu | Intermedju ta' Sitagliptin Phosphate Monohydrate (CAS: 654671-77-9) |
Pakkett: Flixkun, borża tal-fojl tal-aluminju, 25kg/Drum tal-Kartun, jew skont il-ħtieġa tal-klijent.
Kundizzjoni tal-Ħżin:Aħżen f'kontenituri ssiġillati f'post frisk u niexef;Ipproteġi mid-dawl u l-umdità.
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2,4,5-Trifluorophenylacetic Acid (CAS: 209995-38-0) huwa intermedju ta 'Sitagliptin Phosphate Monohydrate (CAS: 654671-77-9).Sitagliptin Phosphate (STG) jintuża biex jikkura DM tip 2 minħabba li jtejjeb il-kontroll gliċemiku billi jżid il-livelli ta 'ormoni incretin attivi, GLP-1 (peptide-1) u GIP (peptide insulinotropiku dipendenti fuq il-glukożju).L-attivazzjoni ta 'dawn l-incretins fiċ-ċelloli β-frixa tikkawża livelli ogħla ta' adenosine monophosphate ċikliku (cAMP) u kalċju intraċellulari, b'sekrezzjoni sussegwenti ta 'insulina dipendenti fuq il-glukożju (2).Din il-mediċina ipogliċemika tappartjeni għal klassi ġdida msejħa inibituri dipeptidyl peptidase IV.STG ġie approvat mill-FDA fl-2006.
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Sitagliptin CAS 486460-32-6 Purità > 99.0% (HPLC...
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Sitagliptin Phosphate Monohydrate CAS 654671-77...
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Aċidu 2,4,5-Trifluorofenilaċetiku CAS 209995-38-...
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Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Buty...
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Sitagliptin Triazole Hydrochloride CAS 762240-9...
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Sitagliptin Phosphate Monohydrate Intermedju...