Sitagliptin Triazole Hydrochloride CAS 762240-92-6 Mama>99.0% (HPLC) Falegaosimea Maualuluga
Tuuina atu le Sitagliptin Phosphate Monohydrate Fesoʻotaʻi Faʻatasi:
Sitagliptin API CAS 486460-32-6
Sitagliptin Phosphate Monohydrate API CAS 654671-77-9
2,4,5-Trifluorophenylacetic Acid CAS 209995-38-0
Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Butyric Acid CAS 486460-00-8
Sitagliptin Triazole Hydrochloride CAS 762240-92-6
Sitagliptin Phosphate Monohydrate Intermediate CAS 486460-21-3
Igoa Vailaau | 3-(Trifluoromethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine Hydrochloride |
Synonyms | Sitagliptin Triazole Hydrochloride;Sitagliptin Intermediate A |
Numera CAS | 762240-92-6 |
CAT Numera | RF-PI1193 |
Tulaga Fa'asoa | I Fa'atauga, Oloa Fua e O'o i Tone |
Fuafua mole | C6H7F3N4·HCl |
Molecular Weight | 228.60 |
Lisi Lisi | 236.0~246.0 ℃ |
Solubility | Solu i le Methanol |
Fa'ailoga | Ruifu Chemical |
Aitema | Fa'amatalaga |
Fa'aaliga | Pa'epa'e i le Pa'u Pa'epa'e Pa'epa'e |
Faailoaina e le HPLC | Ole taimi ole fa'atumauina ole fa'ata'ita'iga e fetaui lelei ma tulaga fa'asino |
Faailoaina e IR | E usitaia |
Ma'imau ile Fa'amago | <0.50% |
Mea Fa'atatau | |
So'o se Fa'aleaga Ta'itasi | <0.50% |
Aofa'i Fa'aleaga | <1.00% |
Metala mamafa | <20ppm |
Mama / Suʻesuʻega Metotia | >99.0% (HPLC) |
Tulaga Su'ega | Enterprise Standard |
Fa'aoga | Vaeluaga ole Sitagliptin Phosphate Monohydrate (CAS: 654671-77-9) |
afifi: Fagu, taga pepa alumini, 25kg / Cardboard Drum, pe tusa ai ma manaoga o tagata faatau.
Tulaga teuina:Teu i totonu o pusa faʻamaufaʻailoga i se nofoaga malulu ma mago;Puipui mai le malamalama ma le susu.
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3-(Trifluoromethyl) -5,6,7,8-tetrahydro-[1,2,4] triazolo [4,3-a] pyrazine Hydrochloride (CAS: 762240-92-6) o se vaeluagalemu ole Sitagliptin Phosphate Monohydrate ( CAS: 654671-77-9), o se fa'atomuga DPP4 filifilia fa'aola-bioavailable lea na maua e ala i le fa'ata'ita'iina o se vasega o inhibitors DPP4 e maua mai i le β-aminoacid.E fa'aitiitia ai le gaioiga o le DPP4 i se faiga faifaipea pe a mae'a le fa'aaogaina e tasi i aso ta'itasi, fa'asaoina le maualuga o le ta'amilosaga o le GIP ma le GLP1 pe a mae'a taumafataga i su'esu'ega ogaoga ma fa'aumiumi ma fa'aitiitia le maualuga o le kulukose toto e aunoa ma se fa'atuputeleina o le ma'i suka.Sitagliptin Phosphate (STG) e faʻaaogaina e togafitia ai le DM ituaiga 2 aua e faʻaleleia ai le glycemic control e ala i le faʻateleina o le maualuga o hormones incretin, GLP-1 (peptide-1) ma le GIP (glucose-dependent insulinotropic peptide).STG na faʻamaonia e le FDA i le 2006.
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Sitagliptin CAS 486460-32-6 Mama>99.0% (HPLC...
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Sitagliptin Phosphate Monohydrate CAS 654671-77...
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2,4,5-Trifluorophenylacetic Acid CAS 209995-38-...
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Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Buty...
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Sitagliptin Triazole Hydrochloride CAS 762240-9...
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Sitagliptin Phosphate Monohydrate Intermediate ...