Cetrorelix Acetate CAS 130143-01-0 GnRH Antagonist Peptide Purity (HPLC) ≥98.0% Boleng bo Phahameng
Shanghai Ruifu Chemical Co., Ltd. ke moetsi ea ka sehloohong oa Cetrorelix Acetate (CAS: 130143-01-0) e nang le boleng bo phahameng.Cetrorelix Acetate ke mohanyetsi oa gonadotropin-release hormone (GnRH).Ruifu Chemical e fana ka letoto la li-peptide tsa GMP.Ruifu e ka fana ka lits'ebeletso tsa lefats'e ka bophara, theko ea tlholisano, palo e nyane le e ngata e fumanehang.Reka Cetrorelix Acetate,Please contact: alvin@ruifuchem.com
Lebitso la Lik'hemik'hale | Cetrorelix Acetate |
Litlhaloso tse tšoanang | N-Acetyl-3-(2-Naphthalenyl)-D-Alanyl-4-Chloro-D-Phenylalanyl-3-(3-Pyridinyl)-D-Alanyl-L-Seryl-L-Tyrosyl-N5-(Aminocarbonyl)- D-Ornithyl-L-Leucyl-L-Arginyl-L-Prolyl-D-Alaninamide Diacetate;NS-75A Diacetate;SB-075 Diacetate |
Tatelano | Ac-3-(2-naphthyl)-D-Ala-4-Chloro-D-Phe-3(3-pyridyl)-D-Ala-Ser-Tyr-D-Cit-Leu-Arg-Pro-D-Ala -NH2 |
Nomoro ea CAS | 130143-01-0 |
Boemo ba Setoko | Ka Setokong, Sekhahla sa Tlhahiso Ho fihlela ho Lik'hilograma |
Foromo ea limolek'hule | Setšoantšo sa C70H92N17O14 |
Boima ba Molek'hule | 1551.16 |
Mocheso oa polokelo. | Sebaka se pholileng le se omileng (-20℃).Sehatsetsi |
Shelf Life | > Lilemo tse 2 haeba li bolokiloe hantle |
Sehlopha | Li-peptide tsa GMP |
Tokomane | COA, MS, HPLC, NMR, MSDS, joalo-joalo. |
Brand | Ruifu Chemical |
Ntho | Litlhaloso |
Ponahalo | Phofo e Tshweu |
Peptide Purity (ka HPLC) | ≥98.0% (ka Area Integration) |
Litaba tsa Peptide | ≥80.0% (ka %N) |
Sebopeho sa Amino Acid | 10% ea Theetical |
Litaba tsa Acetate | ≤10.0% (ka HPLC) |
Litaba tsa TFA | ≤1.0% |
Tšilafalo e le Mong | ≤1.0% (ka HPLC) |
Litaba tsa Metsi (Karl Fischer) | ≤8.0% |
Tlhahlobo | 95.0~105.0% (Ka Anhydrous, Acetic-Free) |
MS | E tsitsitseng |
Tekanyetso ea Teko | Maemo a Khoebo |
Litlhoko tsa ho Romela | Mekotla ea leqhoa, Mekotla ea Desiccant |
Tšimoloho ea Sehlahisoa | Synthetic |
Tlhokomeliso | Feela Bakeng sa Lipatlisiso, Eseng Bakeng sa Tšebeliso ea Batho |
Tšebeliso | Mohanyetsi oa Synthetic oa Moamoheli oa GnRH |
Sephutheloana:Vial ea polasetiki (e nehetsoeng ho paka peptide) kapa vial ea khalase, bongata ho latela tlhoko ea lintlha tsa moreki.
Boemo ba polokelo:Boloka ka lijaneng tse tiisitsoeng sebakeng sa polokelo se pholileng le se omileng (2~8℃) hole le lintho tse sa lumellaneng.Sireletsa leseli le mongobo.
Ho tsamaisa ka sekepe:Fana ka lefatše ka FedEx / DHL Express.Fana ka thomello e potlakileng le e tšepahalang.
Cetrorelix Acetate (CAS 130143-01-0) ke mohanyetsi oa gonadotropin-releasing hormone (GnRH) e rekisoang haholo-holo tlas'a lebitso la Cetrotide.Decapeptide ea maiketsetso, e sebelisoa ho thusa ho tsoala ho thibela ho eketseha ha lihomone tsa luteinizing pele ho nako.Setlhare sena se sebetsa ka ho thibela ketso ea GnRH holim'a pituitary, kahoo e thibela ka potlako tlhahiso le ketso ea hormone ea luteinizing (LH) le follicle-stimulating hormone (FSH).Cetrorelix Acetate e entsoe ka mefuta e fapaneng ea li-amino acid tseo e seng tsa tlhaho tse thibelang ho hlaha ha mahe pele ho liteko tsa bongaka, tse lebisang pokellong ea ovulation le ho thusa kalafo ea theknoloji ea ho ikatisa bakeng sa bakuli ba nang le ts'usumetso e laoloang ea mahe a bomme.
Pontšo Cetrorelix Acetate ke hormone ea maiketsetso e thibelang liphello tsa gonadotropin-releasing hormone (GnRH).Ho thekenoloji e thusang ea ho ikatisa, ho bakuli ba nang le ts'usumetso e laoloang ea mae a bomme, thibela ho tsoa pele ho nako.
Ketso ea Pharmacological Cetrorelix Acetate ke mohanyetsi oa gonadotropin-release hormone (GnRH).GnRH e ka tlama ho li-membrane receptors tsa lisele tsa pituitary.Cetrorelix acetate e tlama ka tlholisano ho li-receptor tsena tse nang le GnRH e sa feleng, ka hona e thibela ho hlahisoa ha hormone ea luteinizing (LH) le follicle stimulating hormone (FSH) ka adenohypophysis.Tšusumetso e thibelang e ile ea hlahisoa hang ka mor'a tsamaiso ea cetrorelix acetate, 'me phello ea ho thibela e ka bolokoa ka phekolo e tsoelang pele.bakeng sa basali, Cetrorelix Acetate e ka liehisa tlhōrō ea LH, kahoo e liehisa ovulation.Bakeng sa basali ba nang le ts'usumetso ea mahe a bomme, nako ea ts'ebetso e ne e itšetlehile ka tekanyo.Tekanyo e le 'ngoe ea cetrorelix 3mg e ne e hakanngoa hore e na le phello e thibelang bonyane matsatsi a 4, e nang le phello e thibelang hoo e ka bang 70% ka Letsatsi la 4. Tsamaiso e pheta-phetoang ea cetrorelix acetate 0.25mg lihora tse ling le tse ling tsa 24 e ka boloka phello ea eona.Phello e hanyetsang li-hormone ea Cetrorelix Acetate e ile ea fetoha ka ho feletseng qetellong ea phekolo ho liphoofolo le batho.
Mosebetsi oa likokoana-hloko Cetrorelix Acetate ke mohanyetsi ea matla oa mokelikeli oa GnRH ea nang le boleng ba IC50 ba 1.21 nM.
Sepheo sa IC50: 1.21 nM GnRH.