Sitagliptin CAS 486460-32-6 Mimo>99.0% (HPLC) API Iwa Mimo giga
Ipese Sitagliptin Phosphate Monohydrate Awọn agbedemeji ibatan:
Sitagliptin API CAS 486460-32-6
Sitagliptin Phosphate Monohydrate API CAS 654671-77-9
2,4,5-Trifluorophenylacetic Acid CAS 209995-38-0
Boc-(R) -3-Amino-4- (2,4,5-Trifluoro-Phenyl) -Butyric Acid CAS 486460-00-8
Sitagliptin Triazole Hydrochloride CAS 762240-92-6
Sitagliptin Phosphate Monohydrate Agbedemeji CAS 486460-21-3
Orukọ Kemikali | Sitagliptin |
Awọn itumọ ọrọ sisọ | (3R) -3-Amino-1- [3- (trifluoromethyl) -5,6,7,8-tetrahydro-1,2,4-triazolo [4,3-a] pyrazin-7-yl] -4- (2,4,5-trifluorophenyl) butan-1-ọkan |
Nọmba CAS | 486460-32-6 |
Iṣura Ipo | Ninu Iṣura, Iwọn iṣelọpọ Ti o to Awọn Toonu |
Fọọmu Molecular | C16H15F6N5O |
Òṣuwọn Molikula | 407.31 |
Ojuami Iyo | 114.0 ~ 115.0 ℃ |
Brand | Ruifu Kemikali |
Nkan | Awọn pato |
Ifarahan | Funfun lati Pa-White Crystalline Powder |
Idanimọ nipa HPLC | Akoko Idaduro ti Ayẹwo jẹ Concordant Pẹlu Iwọn Itọkasi |
Pipadanu lori Gbigbe | <1.0% |
Aloku lori Iginisonu | <0.20% |
Awọn nkan ti o jọmọ | |
Eyikeyi Nikan Aimọ | <0.50% |
Lapapọ Awọn Aimọ | <1.0% |
Mimo | > 99.0% (HPLC) |
Enantiomeric ti nw | <0.50% |
Awọn irin Heavy | <20ppm |
Igbeyewo Standard | Standard Enterprise |
Lilo | API;Iru II Àtọgbẹ mellitus |
Package: Igo, apo apamọwọ Aluminiomu, 25kg / Paali Drum, tabi gẹgẹbi ibeere alabara.
Ipò Ìpamọ́:Fipamọ sinu awọn apoti ti a fi edidi ni itura ati ibi gbigbẹ;Dabobo lati ina ati ọrinrin.
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Sitagliptin (CAS: 486460-32-6), bii iru oogun antidiabetic tuntun, Sitagliptin Phosphate ni awọn anfani ti igbẹkẹle glukosi, ipa hypoglycemic iwọntunwọnsi, yomijade pọ si laisi hypoglycemia, dinku ebi ni imunadoko, ati pe ko ni awọn ipa ẹgbẹ bii ríru, ìgbagbogbo, edema ati iwuwo ara ti o pọ sii.Sitagliptin fosifeti gẹgẹbi itọju oogun kan ni awọn alaisan ti o ni àtọgbẹ iru II le dinku ipele haemoglobin glycosylated (HbA1c) ni pataki.O jẹ dipeptidyl peptidase-4 (DPP-4) inhibitor, eyiti o le mu agbara ara eniyan dara lati dinku ipele glukosi ẹjẹ giga.Sitagliptin jẹ idagbasoke nipasẹ Merck & Co. ati fọwọsi fun lilo iṣoogun ni Amẹrika ni ọdun 2006.
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Sitagliptin CAS 486460-32-6 Mimọ>99.0% (HPLC...
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Sitagliptin Phosphate Monohydrate CAS 654671-77...
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2,4,5-Trifluorophenylacetic Acid CAS 209995-38-...
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Boc-(R) -3-Amino-4- (2,4,5-Trifluoro-Phenyl)-Buty...
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Sitagliptin Triazole Hydrochloride CAS 762240-9...
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Sitagliptin Phosphate Monohydrate Agbedemeji ...