I-Cetrorelix Acetate CAS 130143-01-0 GnRH Antagonist Peptide Purity (HPLC) ≥98.0% Isithombe Esifakiwe Sekhwalithi Ephezulu

I-Cetrorelix Acetate CAS 130143-01-0 GnRH Antagonist Peptide Purity (HPLC) ≥98.0% Ikhwalithi ephezulu

Incazelo emfushane:

Igama Lekhemikhali: I-Cetrorelix Acetate

I-CAS: 130143-01-0

Ukubukeka: Impushana Emhlophe

I-Peptide Purity (HPLC): ≥98.0%

I-Synthetic Antagonist ye-GnRH Receptor

GMP Peptides, API, High Quality

Thintana: UDkt. Alvin Huang

Iselula/Wechat/WhatsApp: +86-15026746401

E-Mail: alvin@ruifuchem.com

Thumela i-imeyili kithi

Imininingwane Yomkhiqizo

Imikhiqizo Ehlobene

Omaka bomkhiqizo

Incazelo:

I-Shanghai Ruifu Chemical Co., Ltd. ingumkhiqizi ohamba phambili we-Cetrorelix Acetate (CAS: 130143-01-0) enekhwalithi ephezulu.I-Cetrorelix Acetate imelene ne-gonadotropin-releasing hormone (GnRH).I-Ruifu Chemical ihlinzeka ngochungechunge lwama-peptide e-GMP.I-Ruifu inganikeza ukulethwa komhlaba wonke, intengo encintisanayo, amanani amancane nayinqwaba atholakalayo.Thenga i-Cetrorelix Acetate,Please contact: alvin@ruifuchem.com

Chemical Properties:

Igama Lekhemikhali	I-Cetrorelix Acetate
Omqondofana	N-Acetyl-3-(2-Naphthalenyl)-D-Alanyl-4-Chloro-D-Phenylalanyl-3-(3-Pyridinyl)-D-Alanyl-L-Seryl-L-Tyrosyl-N5-(Aminocarbonyl)- I-D-Ornithyl-L-Leucyl-L-Arginyl-L-Prolyl-D-Alaninamide Diacetate;I-NS-75A Diacetate;I-SB-075 Diacetate
Ukulandelana	Ac-3-(2-naphthyl)-D-Ala-4-Chloro-D-Phe-3(3-pyridyl)-D-Ala-Ser-Tyr-D-Cit-Leu-Arg-Pro-D-Ala -NH2
Inombolo ye-CAS	130143-01-0
Isimo Sesitoko	Esitokweni, Isikali Sokukhiqiza Sifinyelela Kumakhilogremu
I-Molecular Formula	I-C70H92N17O14
Isisindo samangqamuzana	1551.16
Isikhathi Sokugcina.	Indawo Epholile Neyomile (-20℃).Isiqandisi
I-Shelf Life	> Iminyaka engu-2 uma Igcinwe Kahle
Isigaba	GMP Peptides
Idokhumenti	I-COA, MS, HPLC, NMR, MSDS, njll.
Ibhrendi	I-Ruifu Chemical

Imininingwane:

Into	Imininingwane
Ukubukeka	Impushana Emhlophe
I-Peptide Purity (nge-HPLC)	≥98.0% (nge-Area Integration)
Okuqukethwe kwe-Peptide	≥80.0% (ngo-%N)
Ukwakhiwa kwe-Amino Acid	I-10% ye-Theetical
Okuqukethwe kwe-Acetate	≤10.0% (nge-HPLC)
Okuqukethwe kwe-TFA	≤1.0%
Ukungcola Okukodwa	≤1.0% (nge-HPLC)
Okuqukethwe kwamanzi (Karl Fischer)	≤8.0%
Isivivinyo	95.0~105.0% (Nge-Anhydrous, I-Acetic-Free)
MS	Kuyavumelana
Izinga Lokuhlola	I-Enterprise Standard
Izidingo Zokuthumela	Izikhwama zeqhwa, Izikhwama zeDesiccant
Umsuka Womkhiqizo	Zokwenziwa
Ukunaka	Okokucwaninga Kuphela, Hhayi Okokusetshenziswa Komuntu
Ukusetshenziswa	I-Synthetic Antagonist ye-GnRH Receptor

Iphakheji nesitoreji:

Iphakheji:Isitsha sepulasitiki (esinikezelwe ukupakisha i-peptide) noma isitsha sengilazi, ubuningi ngokuya ngesidingo semininingwane yekhasimende.
Isimo Sesitoreji:Gcina ezitsheni ezivaliwe endaweni epholile neyomile (2~8℃) kude nezinto ezingahambelani.Vikela ekukhanyeni nakumswakama.
Ukuthumela:Thumela emhlabeni wonke nge-FedEx / DHL Express.Nikeza ukulethwa okusheshayo nokuthembekile.

Izinzuzo:

I-FAQ:

Isicelo:

I-Cetrorelix Acetate (CAS 130143-01-0) iyimbangi ye-gonadotropin-releasing hormone (GnRH) ethengiswa kakhulukazi ngaphansi kwegama lomkhiqizo elithi Cetrotide.I-decapeptide yokwenziwa, isetshenziswa ekusizeni ukukhiqiza kabusha ukuvimbela ukukhuphuka kwe-hormone ye-luteinizing ngaphambi kwesikhathi.Umuthi usebenza ngokuvimbela isenzo se-GnRH phezu kwe-pituitary, ngaleyo ndlela ucindezele ngokushesha ukukhiqizwa nokusebenza kwe-hormone ye-luteinizing (LH) kanye ne-follicle-stimulating hormone (FSH).I-Cetrorelix Acetate yenziwe ngezinhlobonhlobo zama-amino acid angewona awemvelo avimbela ukuphuma kweqanda kwangaphambi kwesikhathi ezivivinyweni zomtholampilo, okuholela ekuqoqweni kwe-ovulation kanye nokwelashwa kobuchwepheshe bokuzala okusizwayo ezigulini ezilawulwa yi-ovarian stimulation.
Inkomba i-Cetrorelix Acetate iyi-hormone yokwenziwa evimba imiphumela ye-gonadotropin-releasing hormone (GnRH).Kubuchwepheshe bokusiza bokuzala, ezigulini ezilawulwa yi-ovarian stimulation, vimbela ukuvuthwa ngaphambi kwesikhathi.
Isenzo se-Pharmacological I-Cetrorelix Acetate imelene ne-gonadotropin-releasing hormone (GnRH).I-GnRH ingabophezela kuma-membrane receptors amaseli e-pituitary.I-Cetrorelix acetate ibophezela ngokuncintisana kulawa ma-receptors ane-GnRH engapheli, ngaleyo ndlela ivimbele ngokuncika umthamo we-luteinizing hormone (LH) kanye ne-follicle stimulating hormone (FSH) nge-adenohypophysis.Umphumela ovimbelayo wakhiqizwa ngokushesha ngemva kokuphathwa kwe-cetrorelix acetate, futhi umphumela wokuvimbela ungagcinwa ngokwelashwa okuqhubekayo.kwabesifazane, i-Cetrorelix Acetate ingabambezela ukuphakama kwe-LH, ngaleyo ndlela ibambezele i-ovulation.Kwabesifazane abathola ukugqugquzelwa kwe-ovarian, ubude besenzo babuncike kumthamo.Umthamo owodwa we-cetrorelix 3mg kulinganiselwa ukuthi unomphumela wokuvimbela okungenani izinsuku ezingu-4, nomphumela wokuvimbela cishe we-70% ngosuku lwe-4. Ukuphathwa okuphindaphindiwe kwe-cetrorelix acetate 0.25mg njalo amahora angu-24 kungagcina umphumela wawo.Umphumela we-hormone-antagonizing we-Cetrorelix Acetate wahlehliswa ngokuphelele ekupheleni kokwelashwa ezilwaneni nakubantu.
Umsebenzi webhayoloji i-Cetrorelix Acetate iwumbangi onamandla wesamukeli se-GnRH enevelu ye-IC50 engu-1.21 nM.
Ithagethi IC50: 1.21 nM GnRH.