I-Sitagliptin CAS 486460-32-6 Purity >99.0% (HPLC) API Factory High Purity
Thola Izimo Ezihlobene Ne-Sitagliptin Phosphate Monohydrate:
I-Sitagliptin API CAS 486460-32-6
I-Sitagliptin Phosphate Monohydrate API CAS 654671-77-9
2,4,5-Trifluorophenylacetic Acid CAS 209995-38-0
I-Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Butyric Acid CAS 486460-00-8
I-Sitagliptin Triazole Hydrochloride CAS 762240-92-6
I-Sitagliptin Phosphate Monohydrate Intermediate CAS 486460-21-3
Igama Lekhemikhali | I-Sitagliptin |
Omqondofana | (3R)-3-Amino-1-[3-(trifluoromethyl)-5,6,7,8-tetrahydro-1,2,4-triazolo[4,3-a]pyrazin-7-yl]-4- (2,4,5-trifluorophenyl)butan-1-one |
Inombolo ye-CAS | 486460-32-6 |
Isimo Sesitoko | Esitokweni, Isikali Sokukhiqiza Sifinyelela Kumathani |
I-Molecular Formula | I-C16H15F6N5O |
Isisindo samangqamuzana | 407.31 |
I-Melting Point | 114.0~115.0℃ |
Ibhrendi | I-Ruifu Chemical |
Into | Imininingwane |
Ukubukeka | I-Crystalline Powder emhlophe ukuya kokumhlophe |
Ukuhlonza nge-HPLC | Isikhathi Sokugcina Sesampula Sihambisana Nezithenjwa Ezijwayelekile |
Ukulahlekelwa Ekumisweni | <1.0% |
Izinsalela ekushiseni | <0.20% |
Izinto Ezihlobene | |
Noma Ikuphi Ukungcola Okukodwa | <0.50% |
Ukungcola Okuphelele | <1.0% |
Ubumsulwa | >99.0% (HPLC) |
I-Enantiomeric Purity | <0.50% |
Izinsimbi Ezisindayo | <20ppm |
Izinga Lokuhlola | I-Enterprise Standard |
Ukusetshenziswa | I-API;Uhlobo II sikashukela i-mellitus |
Iphakheji: Ibhodlela, isikhwama se-Aluminium foil, 25kg/Cardboard Drum, noma ngokwezidingo zekhasimende.
Isimo Sesitoreji:Gcina ezitsheni ezivaliwe endaweni epholile neyomile;Vikela ekukhanyeni nakumswakama.
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I-Sitagliptin (CAS: 486460-32-6), njengohlobo olusha lomuthi we-antidiabetic, i-Sitagliptin Phosphate inezinzuzo zokuncika kushukela, umphumela olinganiselayo we-hypoglycemic, ukwanda kokukhiqizwa ngaphandle kwe-hypoglycemia, idambise indlala ngempumelelo, futhi ayinayo imiphumela emibi efana nesicanucanu, ukuhlanza, i-edema nokwanda kwesisindo somzimba.I-Sitagliptin phosphate njengomuthi owodwa wokwelashwa ezigulini ezinesifo sikashukela sohlobo II inganciphisa kakhulu izinga le-glycosylated hemoglobin (HbA1c).Kuyi-dipeptidyl peptidase-4 (DPP-4) inhibitor, engathuthukisa ikhono lomzimba womuntu lokwehlisa izinga le-glucose ephezulu egazini.I-Sitagliptin yathuthukiswa ngabakwa-Merck & Co. futhi yagunyazwa ukusetshenziswa kwezokwelapha e-United States ngo-2006.
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I-Sitagliptin CAS 486460-32-6 Ubumsulwa >99.0% (HPLC...
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I-Sitagliptin Phosphate Monohydrate CAS 654671-77...
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2,4,5-Trifluorophenylacetic Acid CAS 209995-38-...
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I-Boc-(R)-3-Amino-4-(2,4,5-Trifluoro-Phenyl)-Buty...
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I-Sitagliptin Triazole Hydrochloride CAS 762240-9...
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I-Sitagliptin Phosphate Monohydrate Intermediate ...